SCHEMBL6053176

SCHEMBL6053176

O=C(c1ccc(-c2ccccc2)c(C(F)(F)F)c1)N1CCC[C@H]1CN1CCCC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.54
HRH3 Q9Y5N1 12/20 0.52
PDK2 Q15119 1/20 0.52
ALK Q9UM73 2/20 0.49
FFAR2 O15552 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2345865 0.88 MET (0.60) METHRH3PDK2ALKKCNH2
SCHEMBL2345863 0.88 MET (0.60) METHRH3PDK2ALKKCNH2
SCHEMBL2344325 0.81 HRH3 (0.65) METHRH3ALKKCNH2
SCHEMBL2344330 0.81 HRH3 (0.65) METHRH3ALKKCNH2
SCHEMBL2403402 0.80 HRH3 (0.54) METHRH3ALKKCNH2
SCHEMBL2340660 0.79 MET (0.61) METHRH3ALKKCNH2
SCHEMBL12393031 0.79 MET (0.61) METHRH3ALKKCNH2
Trifluoroacetic Acid SCHEMBL2340746 0.79 ALK (0.58) METHRH3PDK2ALKKCNH2
Trifluoroacetic Acid SCHEMBL2340751 0.79 ALK (0.58) METHRH3PDK2ALKKCNH2
SCHEMBL10293596 0.78 HRH3 (0.62) METHRH3ALKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735278-A1 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND THERAPEUTIC USES ELI LILLY AND COMPANY (US) 2006-12-27 EP disclosed
WO-2005097740-A1 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND THERAPEUTIC USES ELI LILLY AND COMPANY (US) 2005-10-20 WO disclosed