SCHEMBL6061201

SCHEMBL6061201

CCOC(=O)c1c(CC(O)N(C)C(=O)OCc2ccccc2)c2ncc(Cc3ccc(F)cc3)cc2[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
ALOX5 P09917 1/20 0.37
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
CCR6 P51684 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5A P29375 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6061617 0.93 NPC1 (0.36) NPC1RAB9AALOX5KMT2AKDM4E
SCHEMBL4761738 0.76 KDM5A (0.52) NPC1RAB9AALOX5KMT2AKDM4E
SCHEMBL6061670 0.76 KDM5A (0.39) NPC1RAB9AALOX5KMT2AKDM4E
SCHEMBL6061005 0.76 KDM5A (0.38) NPC1RAB9AALOX5KMT2AKDM4E
SCHEMBL4297249 0.74 KDM5A (0.54) ALOX5KDM4EMAPTKDM5AKDM5B
SCHEMBL6061157 0.72 ALOX5 (0.37) NPC1RAB9AALOX5KMT2AKDM4E
SCHEMBL15163676 0.71 BRS3 (0.35) KMT2AKDM4EMEN1TDP1
SCHEMBL27666982 0.71 BTK (0.34) KMT2AKDM4EMEN1TDP1
SCHEMBL27686061 0.71 TDP1 (0.36) TDP1
SCHEMBL6061268 0.70 GAA (0.37) NPC1RAB9AALOX5KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720856-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-15 EP disclosed
WO-2005077050-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-25 WO disclosed