SCHEMBL6061670

SCHEMBL6061670

CCOC(=O)c1c(CCC(O)S(C)(=O)=O)c2ncc(Cc3ccc(F)cc3)cc2[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
CCR6 P51684 1/20 0.38
KMT2A Q03164 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALOX5 P09917 1/20 0.37
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
MAP3K5 Q99683 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6061005 0.86 KDM5A (0.38) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL6061617 0.81 NPC1 (0.36) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL4761738 0.81 KDM5A (0.52) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL27667170 0.77 BTK (0.33) KDM4EMEN1KMT2A
SCHEMBL6061201 0.76 NPC1 (0.37) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL6061253 0.74 TDP1 (0.34) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL6061268 0.74 GAA (0.37) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL6061157 0.73 ALOX5 (0.37) KDM5AKDM5BKDM4EMEN1ALDH1A1
SCHEMBL5545516 0.72 KDM5A (0.47) KDM5AKDM5BKDM4EALDH1A1LMNA
SCHEMBL27686061 0.71 TDP1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720856-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-15 EP disclosed
WO-2005077050-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-25 WO disclosed