SCHEMBL6064058

SCHEMBL6064058

OC(Cc1ccccc1)N1CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.61
CYP2C19 P33261 6/20 0.61
CYP3A4 P08684 5/20 0.61
CYP2D6 P10635 5/20 0.61
TSHR P16473 4/20 0.61
RAB9A P51151 1/20 0.50
KCNA5 P22460 7/20 0.47
CYP2C9 P11712 5/20 0.47
KCNH2 Q12809 4/20 0.47
KCNE1 P15382 2/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HPGD P15428 3/20 0.46
GAA P10253 2/20 0.46
SIGMAR1 Q99720 1/20 0.44
IDO1 P14902 1/20 0.44
LMNA P02545 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL583721 0.98 CYP1A2 (0.58) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
Hydrochloric Acid SCHEMBL8017800 0.96 CYP1A2 (0.56) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL4131831 0.81 SLC6A4 (0.63) SIGMAR1KMT2A
SCHEMBL8125629 0.81 ALDH1A1 (0.50) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL10454919 0.81 KCNA5 (0.49) TSHRKCNA5KCNH2GAASIGMAR1
SCHEMBL27364544 0.79 SIGMAR1 (0.50) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL7213383 0.78 IDO1 (0.71) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL465921 0.78 KCNA5 (0.62) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL6889456 0.77 KMT2A (0.62) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL6479214 0.77 CYP1A2 (0.61) CYP1A2CYP2C19CYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105237467-B A kind of preparation method of doxylamine succinate 南京济群医药科技股份有限公司 2017-12-08 CN claimed
US-7087549-B2 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY (US) 2006-08-08 US claimed
US-20050181935-A1 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY 2005-08-18 US claimed
EP-0990670-B1 Calcium-based catalyst system GOODYEAR TIRE & RUBBER (US) 2004-11-03 EP claimed
US-20020045720-A1 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY 2002-04-18 US claimed
US-6359088-B1 COPOLYMERIZING STYRENE AND 1,3-BUTADIENE IN AN ORGANIC SOLVENT IN THE PRESENCE OF CATALYST SYSTEM WHICH CONSISTS ESSENTIALLY OF AN ORGANOLITHIUM COMPOUND, A CALCIUM ALKOXIDE AND A LITHIUM ALKOXIDE THE GOODYEAR TIRE & RUBBER COMPANY 2002-03-19 US claimed
US-6103842-A USING CATALYST SYSTEM FOR EXOTHERMAL POLYMERIZATION WHICH CONSISTS ESSENTIALLY OF (A) AN ORGANOLITHIUM COMPOUND, (B) A BARIUM ALKOXIDE AND (C) A LITHIUM ALKOXIDE THE GOODYEAR TIRE & RUBBER COMPANY (US) 2000-08-15 US claimed
EP-0990670-A1 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY (US) 2000-04-05 EP claimed
EP-0391692-B1 Process for producing high trans low vinyl conjugated diene (co) polymer JAPAN SYNTHETIC RUBBER CO LTD (JP) 1994-01-05 EP claimed
US-5086136-A Using coordination catalyst containing organoaluminum compound, barium compound and alcohol JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1992-02-04 US claimed
EP-0391692-A1 Process for producing high trans low vinyl conjugated diene (co) polymer JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1990-10-10 EP claimed
CN-107056685-A Method for synthesizing doxylamine succinate 珠海市海瑞德生物科技有限公司 2017-08-18 CN disclosed
US-7087549-B2 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY (US) 2006-08-08 US disclosed
US-20050181935-A1 Calcium-based catalyst system THE GOODYEAR TIRE & RUBBER COMPANY 2005-08-18 US disclosed
EP-0990670-B1 Calcium-based catalyst system GOODYEAR TIRE & RUBBER (US) 2004-11-03 EP disclosed
US-5086136-A Using coordination catalyst containing organoaluminum compound, barium compound and alcohol JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1992-02-04 US disclosed
EP-0331400-B1 CATALYST COMPOSITION FOR POLYMERIZATION OF CONJUGATED DIENE AND PROCESS FOR PRODUCING CONJUGATED DIENE POLYMER JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1992-01-08 EP disclosed
EP-0391692-A1 Process for producing high trans low vinyl conjugated diene (co) polymer JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1990-10-10 EP disclosed
US-4933401-A ORGANO-LITHIUM-ALUMINUM COMPOUND JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1990-06-12 US disclosed
EP-0331400-A1 Catalyst composition for polymerization of conjugated diene and process for producing conjugated diene polymer JAPAN SYNTHETIC RUBBER CO., LTD. (JP) 1989-09-06 EP disclosed