SCHEMBL6065704

SCHEMBL6065704

CCOC(=O)Cc1c[nH]c2cc(OCc3c(C)c(-c4ccc(Cl)cc4)nn3C)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.43
PPARG P37231 2/20 0.39
MAPT P10636 5/20 0.38
LMNA P02545 4/20 0.38
TP53 P04637 3/20 0.38
THRB P10828 1/20 0.38
SLC2A2 P11168 1/20 0.37
KDM4E B2RXH2 5/20 0.37
KMT2A Q03164 5/20 0.37
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 4/20 0.37
TDP1 Q9NUW8 1/20 0.37
SLC34A1 Q06495 1/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 2/20 0.36
TSHR P16473 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.35
ICMT O60725 1/20 0.35
HPGD P15428 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6064619 0.91 PPARG (0.42) PPARGMAPTLMNATP53KDM4E
SCHEMBL6065163 0.90 PKM (0.41) PKMPPARGSLC34A1
SCHEMBL6064586 0.82 PPARG (0.42) PPARGMAPTLMNATP53THRB
SCHEMBL6065357 0.82 PKM (0.40) PKMPPARGSLC34A1
SCHEMBL6065157 0.80 PPARD (0.45) PPARG
SCHEMBL6064601 0.78 PKM (0.43) PKMMAPTLMNATP53KMT2A
SCHEMBL6065143 0.74 PKM (0.42) PKMMAPTALDH1A1TDP1SLC34A1
SCHEMBL6064609 0.74 PKM (0.42) PKMPPARGMAPTPOLB
SCHEMBL6065741 0.74 PKM (0.40) PKMTHRBTDP1ICMT
SCHEMBL6064613 0.73 PPARG (0.40) PPARGMAPTLMNARAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725546-A1 PYRAZOLYL INDOLYL DERIVATIVES AS PPAR ACTIVATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-29 EP disclosed
WO-2005085235-A1 PYRAZOLYL INDOLYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-09-15 WO disclosed