SCHEMBL6064609

SCHEMBL6064609

CCOC(=O)Cc1c[nH]c2cc(OCc3cc(-c4ccc(C(F)(F)F)cc4)nn3C)ccc12

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
PPARD Q03181 10/20 0.38
PPARA Q07869 7/20 0.38
AGER Q15109 1/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
MAOB P27338 1/20 0.36
PPARG P37231 1/20 0.35
FFAR1 O14842 1/20 0.35
PTGS2 P35354 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6065376 0.92 PKM (0.41) PKMPPARDPPARAAGERPOLB
SCHEMBL6065143 0.92 PKM (0.42) PKMPPARDPOLBMAPTFFAR1
SCHEMBL6065379 0.91 PKM (0.40) PKMPPARDPPARAAGERPOLB
SCHEMBL6064615 0.90 PPARD (0.45) PPARDPPARAPPARG
SCHEMBL6065369 0.90 PKM (0.40) PKMPPARDPPARAPOLBMAPT
SCHEMBL6065741 0.90 PKM (0.40) PKMFFAR1SCN9A
SCHEMBL6064601 0.87 PKM (0.43) PKMPOLBMAPTFFAR1SCN9A
SCHEMBL6065163 0.85 PKM (0.41) PKMPPARDPPARAMAOBPPARG
SCHEMBL6065368 0.84 PKM (0.41) PKMPOLBMAPTSCN9A
SCHEMBL6017372 0.84 PKM (0.43) PKMPPARDPPARAMAOBPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725546-A1 PYRAZOLYL INDOLYL DERIVATIVES AS PPAR ACTIVATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-29 EP disclosed
WO-2005085235-A1 PYRAZOLYL INDOLYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-09-15 WO disclosed