SCHEMBL6066286

SCHEMBL6066286

Cc1ccc2c(N3CC[N]CC3)cccc2n1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.60
HTR1A P08908 14/20 0.53
HTR1D P28221 14/20 0.53
HTR1B P28222 14/20 0.53
NCF1 P14598 3/20 0.50
KCNH2 Q12809 8/20 0.49
SLC6A4 P31645 6/20 0.49
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
DRD2 P14416 4/20 0.47
HTR2A P28223 4/20 0.47
HTR7 P34969 4/20 0.47
DRD3 P35462 4/20 0.47
HTR2B P41595 4/20 0.47
HTR6 P50406 1/20 0.47
HTR2C P28335 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10516997 0.87 NCF1 (0.65) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL13525141 0.84 CYP2C9 (0.67) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL428165 0.83 NCF1 (0.69) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL1366345 0.81 NCF1 (0.75) NCF1ADRB2ADRB1
SCHEMBL4178112 0.80 NCF1 (0.59) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL4176462 0.79 NCF1 (0.72) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL3137750 0.75 CYP2C9 (0.50) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL2881010 0.75 CYP2C9 (0.50) CYP2C9HTR1AHTR1DHTR1BNCF1
SCHEMBL13525153 0.75 HTR1A (0.57) CYP2C9HTR1AHTR1DHTR1BKCNH2
SCHEMBL429083 0.75 CYP2C9 (0.50) CYP2C9HTR1AHTR1DHTR1BNCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646613-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES HAVING AFFINITY FOR 5HT1-TYPE RECEPTORS GLAXO GROUP LIMITED (GB) 2006-04-19 EP disclosed
WO-2005014552-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES HAVING AFFINITY FOR 5HT1-TYPE RECEPTORS GLAXO GROUP LIMITED (GB) 2005-02-17 WO disclosed