SCHEMBL6068626

SCHEMBL6068626

O=C1CNCCN1Cc1ccccn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.56
CRBN Q96SW2 1/20 0.56
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 5/20 0.45
MEN1 O00255 1/20 0.45
PKM P14618 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
SLC6A4 P31645 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 2/20 0.42
LMNA P02545 2/20 0.42
OPRM1 P35372 2/20 0.41
P2RX7 Q99572 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30282988 0.81 KDM4E (0.37) DDB1CRBNKMT2ACYP1A2CYP2C19
SCHEMBL21071359 0.80 DDB1 (0.47) DDB1CRBNKMT2ACYP1A2CYP2C19
SCHEMBL13886225 0.79 CXCR4 (0.64) DDB1CRBNALDH1A1L3MBTL1SLC6A4
SCHEMBL92331 0.78 L3MBTL1 (0.56) DDB1CRBNKMT2ACYP2C19ALDH1A1
SCHEMBL4543665 0.78 DDB1 (0.57) DDB1CRBNKMT2ACYP1A2CYP2C19
SCHEMBL27357726 0.77 DDB1 (0.60) DDB1CRBNKMT2ACYP1A2CYP2C19
Bromide SCHEMBL28426487 0.76 L3MBTL1 (0.54) DDB1CRBNKMT2ACYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL4768580 0.76 L3MBTL1 (0.54) DDB1CRBNKMT2ACYP2C19ALDH1A1
SCHEMBL6068660 0.75 DDB1 (0.54) DDB1CRBNKMT2ACYP1A2CYP2C19
SCHEMBL209471 0.74 ALDH1A1 (0.61) DDB1CRBNKMT2ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703765-B Substituted triazole derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2025-02-28 CN disclosed
CN-115703765-A Substituted triazole derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2023-02-17 CN disclosed
WO-2023016521-A1 SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 上海赛默罗生物科技有限公司 2023-02-16 WO disclosed
US-7144887-B2 Substituted 1,2,3-triazolo[1,5-a]quinazolines for enhancing cognition MERCK SHARP & DOHME LTD. (GB) 2006-12-05 US disclosed