SCHEMBL6072979

SCHEMBL6072979

C1=CCN(CCc2sc3ccccc3c2CCc2ccccn2)C1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.45
KCNH2 Q12809 2/20 0.45
CYP2D6 P10635 1/20 0.45
CHRM1 P11229 1/20 0.45
NPY1R P25929 12/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
CASP3 P42574 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072732 0.88 HRH1 (0.58) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6072759 0.88 HRH1 (0.58) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6073337 0.85 HRH1 (0.47) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6072778 0.85 HRH1 (0.43) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6072713 0.82 HRH1 (0.43) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6073196 0.82 NPY1R (0.46) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6072800 0.80 TAS1R3 (0.47) HRH1KCNH2CYP2D6CHRM1NPY1R
SCHEMBL6072802 0.77 HRH3 (0.57) HRH1KCNH2CYP2D6CHRM1TAS1R3
SCHEMBL6072764 0.77 HRH1 (0.65) HRH1KCNH2CYP2D6CHRM1
SCHEMBL4852437 0.74 HRH1 (0.80) HRH1KCNH2CYP2D6CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO claimed
WO-2006019497-A2 SLEEP-INDUCING COMPOUNDS AND METHODS RELATED THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2006-02-23 WO disclosed