SCHEMBL6073650

SCHEMBL6073650

CCCOCCn1c(=O)c(=O)[nH]c2ncc(Br)cc21

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 18/20 0.38
PDE6A P16499 16/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6073334 0.92 ADORA2A (0.39) PDE5APDE6AGRIN1GRIN2B
SCHEMBL20703796 0.85 PDE4D (0.41) PDE6AGRIN1GRIN2B
SCHEMBL6073625 0.84 MEN1 (0.37) PDE5AGRIN1GRIN2B
SCHEMBL6073328 0.79 PDE5A (0.62) PDE5APDE6A
SCHEMBL30635481 0.75 HSD17B10 (0.50)
SCHEMBL1971615 0.75 GRIA1 (0.45) PDE5APDE6AGRIN1GRIN2BKCNH2
SCHEMBL20704356 0.74 PDE4D (0.42) PDE6AGRIN1GRIN2B
SCHEMBL31008703 0.74 GRIN1 (0.58) GRIN1GRIN2B
SCHEMBL20134012 0.74 GRIN1 (0.58) GRIN1GRIN2B
SCHEMBL20704210 0.72 PDE4D (0.48) PDE6AGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006126081-A2 PYRIDINO [2 , 3-B] PYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-11-30 WO disclosed
WO-2006126081-A2 PYRIDINO [2 , 3-B] PYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-11-30 WO disclosed