SCHEMBL6073864

SCHEMBL6073864

CC(=O)N1CCN(c2ccc(Nc3ncc4ccc(NC(=O)NCCCN5CCOCC5)nc4n3)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 3/20 0.50
ALK Q9UM73 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
SYK P43405 12/20 0.46
CDK4 P11802 2/20 0.45
CCND1 P24385 2/20 0.45
CCNE1 P24864 2/20 0.45
CDK2 P24941 2/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6074099 0.89 SMN1; SMN2 (0.46) SMN1; SMN2SYKCDK4CCND1CCNE1
SCHEMBL6073406 0.87 ALK (0.54) ALKSYKCDK4CCND1CCNE1
SCHEMBL6073931 0.86 LMNA (0.53) SMN1; SMN2MAPT
SCHEMBL6074378 0.85 SYK (0.56) JAK3ALKSYKCDK4CCND1
SCHEMBL6074063 0.80 SYK (0.56) JAK3ALKSYKCDK4CCND1
SCHEMBL6073490 0.79 CCND3 (0.50) JAK3ALKSMN1; SMN2SYKCDK4
SCHEMBL6074268 0.78 CDK4 (0.47) JAK3SYKCDK4CCND1CCNE1
SCHEMBL6074659 0.78 SYK (0.58) ALKSYKCDK4CCND1CCNE1
SCHEMBL6074149 0.77 CDK4 (0.46) JAK3SYKCDK4CCND1CCNE1
SCHEMBL6074118 0.76 SYK (0.51) JAK3ALKSYKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030073668-A1 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors BOOTH RICHARD JOHN (US) 2003-04-17 US claimed
EP-1254137-A1 PYRIDO 2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2002-11-06 EP claimed
WO-2001055147-A1 PYRIDO[2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-08-02 WO claimed
US-7053070-B2 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors WARNER-LAMBERT COMPANY (US) 2006-05-30 US disclosed
US-20030073668-A1 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors BOOTH RICHARD JOHN (US) 2003-04-17 US disclosed
EP-1254137-A1 PYRIDO 2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2002-11-06 EP disclosed
WO-2001055147-A1 PYRIDO[2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030073668-A1 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors CDK9, CDK19, CDK3 JAK3 254/4885ALK 457/4885SMN1; SMN2 3957/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.