SCHEMBL6076060

SCHEMBL6076060

COc1ccc(-c2nc3c(c(NC4CCCC4)n2)CCCC3)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
HPGD P15428 2/20 0.51
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.51
MAPT P10636 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
PDE7A Q13946 1/20 0.48
PDE7B Q9NP56 1/20 0.48
USP2 O75604 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
ALOX5 P09917 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6077112 0.99 HPGD (0.50) KDM4EHPGDALDH1A1LMNAMAPT
SCHEMBL5733203 0.98 KDM4E (0.51) KDM4EHPGDALDH1A1LMNAMAPT
SCHEMBL5733788 0.97 HPGD (0.50) KDM4EHPGDALDH1A1LMNAMAPT
SCHEMBL6075985 0.91 FYN (0.46) KDM4EHPGDALDH1A1LMNAMAPT
SCHEMBL6075981 0.91 FYN (0.46) KDM4EHPGDALDH1A1LMNAMAPT
SCHEMBL6075443 0.86 HRH2 (0.47) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL5732453 0.83 ADORA3 (0.46) KDM4EALDH1A1LMNACYP1A2CYP3A4
SCHEMBL5733352 0.82 ADORA3 (0.45) KDM4EALDH1A1LMNAMAPTMEN1
SCHEMBL6076160 0.82 ACP1 (0.45) KDM4EHPGDALDH1A1MAPTALOX5
SCHEMBL6076928 0.81 PDE5A (0.46) KDM4EHPGDALDH1A1MAPTALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045526-B2 Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical preparations comprising them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-05-16 US claimed