SCHEMBL6077447

SCHEMBL6077447

CCO[C@@H](C(=O)NCc1ccc(C#N)cc1N)N1C(=O)c2cccc(F)c2C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.35
BDKRB1 P46663 6/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SLC1A2 P43004 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32
DGAT2 Q96PD7 1/20 0.32
MAP2K1 Q02750 1/20 0.32
ENPP2 Q13822 1/20 0.32
DRD2 P14416 2/20 0.31
DRD3 P35462 1/20 0.31
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6029560 1.00 TNF (0.35) TNFBDKRB1PDE4APDE4BPDE4C
SCHEMBL6029869 0.87 TNF (0.36) TNFBDKRB1KMT2AMEN1
SCHEMBL6029874 0.87 TNF (0.36) TNFBDKRB1KMT2AMEN1
SCHEMBL6029784 0.86 SLC1A2 (0.37) TNFBDKRB1PDE4APDE4BPDE4C
SCHEMBL6029778 0.86 SLC1A2 (0.37) TNFBDKRB1PDE4APDE4BPDE4C
SCHEMBL6078103 0.78 GABRA1 (0.34) TNFDGAT2DRD2DRD3P2RX7
SCHEMBL6078094 0.78 GABRA1 (0.34) TNFDGAT2DRD2DRD3P2RX7
SCHEMBL6076925 0.75 ST14 (0.41)
SCHEMBL6076940 0.75 ST14 (0.41)
SCHEMBL6078428 0.75 F10 (0.38) BDKRB1KMT2ASLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7056932-B2 Heterocyclyl substituted 1-alkoxy acetic acid amides HOFFMAN-LA ROCHE INC. (US) 2006-06-06 US disclosed
US-20050137168-A1 Heterocyclyl substituted 1-alkoxy acetic acid amides HOFFMANN-LA ROCHE INC. 2005-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050137168-A1 Heterocyclyl substituted 1-alkoxy acetic acid amides F12, TFPI, F11 TNF 90/4885BDKRB1 63/4885PDE4A 1358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.