SCHEMBL6077597

SCHEMBL6077597

NC(=O)[C@@H]1CCCN1Cc1cc(F)ccc1-n1cncn1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.45
MAOB P27338 6/20 0.45
GRM2 Q14416 1/20 0.43
SCN3A Q9NY46 1/20 0.41
POLB P06746 1/20 0.41
EGFR P00533 5/20 0.40
LMNA P02545 1/20 0.39
SPHK1 Q9NYA1 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6078064 0.88 F2 (0.47) POLBEGFRSPHK1
SCHEMBL6077686 0.84 MAOA (0.45) MAOAMAOBGRM2SCN3APOLB
SCHEMBL6077730 0.82 F2 (0.39) EGFRIDO1TDO2ALDH1A1
SCHEMBL6920324 0.76 TSHR (0.40)
SCHEMBL6078513 0.74 AAK1 (0.38) POLB
SCHEMBL6078268 0.73 F2 (0.45)
SCHEMBL6919450 0.72 MAOB (0.44) MAOAMAOB
SCHEMBL6914971 0.72 MAOB (0.44) MAOAMAOB
SCHEMBL29586935 0.72 SCN3A (0.49) MAOAMAOBGRM2SCN3APOLB
SCHEMBL6078656 0.71 F2 (0.47) POLBLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7144899-B2 Thrombin inhibitors MERCK & CO., INC. (US) 2006-12-05 US disclosed
US-20040073025-A1 Thrombin inhibitors MERCK SHARP & DOHME CORP. 2004-04-15 US disclosed
WO-2002064559-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040073025-A1 Thrombin inhibitors F2, F11, F10 MAOA 2066/4885MAOB 1593/4885GRM2 4543/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.