SCHEMBL6079371

SCHEMBL6079371

Cc1nc(OC(CCN(C)C(=O)OC(C)(C)C)C(F)(F)F)c(C#N)cc1F

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
GAA P10253 1/20 0.32
RECQL P46063 1/20 0.32
CACNA1G O43497 1/20 0.32
CACNA1B Q00975 1/20 0.32
CACNA1C Q13936 1/20 0.32
HPGD P15428 1/20 0.32
TRPA1 O75762 1/20 0.31
PDK2 Q15119 1/20 0.31
SLC6A4 P31645 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079361 1.00 LMNA (0.36) LMNAALDH1A1GLACYP1A2CYP2C9
SCHEMBL6079017 0.89 CACNA1G (0.31) ALDH1A1GLACACNA1GCACNA1BCACNA1C
SCHEMBL6079011 0.89 CACNA1G (0.31) ALDH1A1GLACACNA1GCACNA1BCACNA1C
SCHEMBL6079148 0.85 SLC6A4 (0.34) ALDH1A1GLACACNA1GCACNA1BCACNA1C
SCHEMBL6078728 0.82 SLC6A4 (0.45) CACNA1GCACNA1BCACNA1CPDK2SLC6A4
SCHEMBL6078732 0.82 SLC6A4 (0.45) CACNA1GCACNA1BCACNA1CPDK2SLC6A4
SCHEMBL6079517 0.76 CACNA1G (0.33) LMNAALDH1A1GLACYP1A2CYP2C9
SCHEMBL6078329 0.75 LMNA (0.38) LMNAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6078323 0.75 LMNA (0.38) LMNAALDH1A1CYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL6078597 0.74 SLC6A4 (0.39) LMNACYP1A2CYP2C9CYP2C19GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119109-B2 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase ASTRAZENECA AB (SE) 2006-10-10 US disclosed