SCHEMBL608221

SCHEMBL608221

FC(F)(F)c1cnc(Cl)cn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.43
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SIRT6 Q8N6T7 1/20 0.35
CA2 P00918 1/20 0.32
CHKA P35790 1/20 0.32
KCNQ3 O43525 2/20 0.32
KCNQ2 O43526 2/20 0.32
KCNE1 P15382 2/20 0.32
KCNQ1 P51787 2/20 0.32
SMARCA2 P51531 1/20 0.32
SMARCA4 P51532 1/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27807873 0.77 SIRT6 (0.41) JUNNFKB1NFKB2RELASIRT6
SCHEMBL18443080 0.76 SIRT6 (0.34) JUNNFKB1NFKB2RELASIRT6
SCHEMBL18442595 0.76 JUN (0.31) JUNNFKB1NFKB2RELASIRT6
SCHEMBL30185867 0.76 SIRT6 (0.34) JUNNFKB1NFKB2RELASIRT6
SCHEMBL9924589 0.75 SIRT6 (0.35) SIRT6
SCHEMBL29770810 0.75 SIRT6 (0.35) SIRT6
SCHEMBL17164929 0.74 SIRT6 (0.41) JUNNFKB1NFKB2RELASIRT6
SCHEMBL933680 0.74
SCHEMBL16635101 0.72 AAK1 (0.39) TRPV4
SCHEMBL17162215 0.72 BACE1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 626 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106499-A1 OREXIN RECEPTOR ANTAGONISTS: 2-AZABICYCLIC COMPOUNDS BIAL - PORTELA & CA., S.A. (PT) 2026-05-21 WO claimed
EP-4688155-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS Bial-Portela & CA, S.A. (PT) 2026-02-11 EP claimed
EP-4688154-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - Portela & Ca., S.A. (PT) 2026-02-11 EP claimed
WO-2025023852-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - PORTELA & CA., S.A. (PT) 2025-01-30 WO claimed
WO-2025023851-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - PORTELA & CA., S.A. (PT) 2025-01-30 WO claimed
CN-107840828-B Synthesis method of 2-chloro-5-trifluoromethylpyrazine 金凯(辽宁)化工有限公司 2020-11-03 CN claimed
CN-108067233-A Improve foam nickel-base catalyst of sludge hot hydrolysis efficiency and preparation method thereof 北京达源环保科技有限公司 2018-05-25 CN claimed
CN-107879583-A Sludge pyrohydrolysis and anaerobic digestion integrated treatment process system 北京达源环保科技有限公司 2018-04-06 CN claimed
CN-107840828-A A kind of synthetic method of the trifluoromethyl pyrazine of 2 chlorine 5 金凯(辽宁)化工有限公司 2018-03-27 CN claimed
CN-101792420-A Preparation of halogenated n-heteroaromatic polyhalogen derivatives SALTIGO GMBH 2010-08-04 CN claimed
WO-2026106499-A1 OREXIN RECEPTOR ANTAGONISTS: 2-AZABICYCLIC COMPOUNDS BIAL - PORTELA & CA., S.A. (PT) 2026-05-21 WO disclosed
US-20260137680-A1 NOVEL COMPOUNDS SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US disclosed
EP-4741018-A2 SULPHONAMIDE COMPOUNDS Anaxis Pharma Pty Ltd (AU) 2026-05-13 EP disclosed
US-12617782-B2 Pyridazinones as PARP7 inhibitors RIBON THERAPEUTICS, INC. (US) 2026-05-05 US disclosed
US-20260085060-A1 THERAPEUTIC COMPOUNDS INDIVIOR UK LTD (GB) 2026-03-26 US disclosed
US-5493024-A 1,2-DIARYL-2-PROPEN-1-ONE CHEMICAL INTERMEDIATE COMPOUND DOWELANCO (US) 1996-02-20 US disclosed
US-5324837-A 3,4-disubstituted-4,5-dihydro-1H-pyrazoles and a method of preparation DOWELANCO (US) 1994-06-28 US disclosed
US-5250532-A Moths. termites DOWELANCO (US) 1993-10-05 US disclosed
CN-1067426-A 3,4, N-three replaces-4,5-dihydro-1 h-pyrazole-1-methane amide and they application as sterilant DOWELANCO (US) 1992-12-30 CN disclosed
EP-0508469-A1 3,4,N-Trisubstituted-4,5-dihydro-1H-pyrazole-1-carboxamides and their use as insecticides DOWELANCO (US) 1992-10-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260137680-A1 NOVEL COMPOUNDS CCR1, CCR4, CCR3 TRPV4 1034/4885JUN 1634/4885NFKB1 293/4885
US-12617782-B2 Pyridazinones as PARP7 inhibitors PARP3, PARP2, PARP1 TRPV4 4429/4885JUN 963/4885NFKB1 4100/4885
US-20260085060-A1 THERAPEUTIC COMPOUNDS HCRTR2, HCRTR1, NPY1R TRPV4 1029/4885JUN 4224/4885NFKB1 1066/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.