SCHEMBL608803

SCHEMBL608803

On1nnc2[c]ccnc21

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2067414 0.76 TP53 (0.32)
SCHEMBL4757736 0.66 MET (0.34)
SCHEMBL3931082 0.65
SCHEMBL34349 0.64 POLB (0.48)
SCHEMBL3943448 0.63
SCHEMBL3934683 0.58
SCHEMBL4059857 0.58
SCHEMBL2067745 0.56
SCHEMBL1190711 0.54
SCHEMBL165149 0.54

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154724-A2 PROCESSES AND COMPOUNDS FOR PREPARING SPIROLIGOMERS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-08-17 WO claimed
US-9695189-B2 Chemical crosslinkers and compositions thereof Nguyen, Mark Quang (US) 2017-07-04 US claimed
US-20140249319-A1 CHEMICAL CROSSLINKERS AND COMPOSITIONS THEREOF Nguyen, Mark Quang (US) 2014-09-04 US claimed
WO-2023154724-A2 PROCESSES AND COMPOUNDS FOR PREPARING SPIROLIGOMERS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-08-17 WO disclosed
US-11111335-B2 Method of preparing carboxylic acid functionalized polymers NEKTAR THERAPEUTICS (US) 2021-09-07 US disclosed
EP-1756173-B1 METHOD OF PREPARING PROPIONIC ACID-TERMINATED POLYMERS NEKTAR THERAPEUTICS (US) 2019-04-03 EP disclosed
US-20180282476-A1 METHOD OF PREPARING CARBOXYLIC ACID FUNCTIONALIZED POLYMERS NEKTAR THERAPEUTICS 2018-10-04 US disclosed
US-10011682-B2 Method of preparing carboxylic acid functionalized polymers NEKTAR THERAPEUTICS (US) 2018-07-03 US disclosed
US-9695189-B2 Chemical crosslinkers and compositions thereof Nguyen, Mark Quang (US) 2017-07-04 US disclosed
EP-2812346-A1 LIGANDS FOR ANTIBODY AND FC-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMOTOGRAPHY IV Graffinity Pharmaceuticals GmbH (DE) 2014-12-17 EP disclosed
US-20140249319-A1 CHEMICAL CROSSLINKERS AND COMPOSITIONS THEREOF Nguyen, Mark Quang (US) 2014-09-04 US disclosed
EP-1692206-B1 METHOD OF PREPARING CARBOXYLIC ACID FUNCTIONALIZED POLYMERS NEKTAR THERAPEUTICS (US) 2010-04-21 EP disclosed
US-20100004428-A1 Method of Preparing Propionic Acid-Terminated Polymers NEKTAR THERAPEUTICS (US) 2010-01-07 US disclosed
US-7608663-B2 reacting a water soluble and non-peptidic polymer comprising at least one hydroxyl group with a tertiary alkyl acrylate in the presence of a catalyst to form a propionic acid ester of the polymer; acid treatment; may be further derivatized; particularly propionic acid-terminated poly(ethylene glycol)s NEKTAR THERAPEUTICS (US) 2009-10-27 US disclosed
EP-1756173-A2 METHOD OF PREPARING PROPIONIC ACID-TERMINATED POLYMERS Nektar Therapeutics Al, Corporation (US) 2007-02-28 EP disclosed
EP-1692206-A1 METHOD OF PREPARING CARBOXYLIC ACID FUNCTIONALIZED POLYMERS Nektar Therapeutics Al, Corporation (US) 2006-08-23 EP disclosed
US-20050214250-A1 Method of preparing carboxylic acid functionalized polymers NEKTAR THERAPEUTICS 2005-09-29 US disclosed
US-20050171291-A1 Method of preparing propionic acid-terminated polymers NEKTAR THERAPEUTICS 2005-08-04 US disclosed
WO-2005070973-A2 METHOD OF PREPARING PROPIONIC ACID-TERMINATED POLYMERS NEKTAR THERAPEUTICS AL, CORPORATION (US) 2005-08-04 WO disclosed
WO-2005047366-A1 METHOD OF PREPARING CARBOXYLIC ACID FUNCTIONALIZED POLYMERS NEKTAR THERAPEUTICS AL, CORPORATION (US) 2005-05-26 WO disclosed