SCHEMBL6089172

SCHEMBL6089172

CC(C)(C)c1cccc(CBr)c1OCC#N

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.35
ALDH1A1 P00352 3/20 0.33
CA2 P00918 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4843386 0.80 SCN4A (0.39) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL6090926 0.80 ALDH1A1 (0.51) NAMPTALDH1A1CA2SMN1; SMN2KDM4E
SCHEMBL22096830 0.78 NAMPT (0.53) NAMPTALDH1A1CA2SMN1; SMN2KDM4E
SCHEMBL9695178 0.77 NR1H4 (0.38) ALDH1A1CA2SMN1; SMN2KDM4E
SCHEMBL6771911 0.73 CA2 (0.34) ALDH1A1CA2SMN1; SMN2KDM4E
SCHEMBL7464494 0.71 PTGER4 (0.33) SMN1; SMN2
SCHEMBL10154387 0.70 CYP1A2 (0.47) NAMPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL3175743 0.68 ALDH1A1 (0.44) ALDH1A1CA2
SCHEMBL27499107 0.68 PTGER4 (0.36) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL9994746 0.66 CA2 (0.61) ALDH1A1CA2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed