SCHEMBL6089640

SCHEMBL6089640

CC(C)OC1=NNC(=O)C1=Cc1cc2c([nH]1)CCCC2=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.39
PDGFRB P09619 7/20 0.36
SRC P12931 6/20 0.36
FGFR1 P11362 5/20 0.36
PKN1 Q16512 1/20 0.35
PKN2 Q16513 1/20 0.35
RET P07949 3/20 0.35
LRRK2 Q5S007 2/20 0.35
ALK Q9UM73 2/20 0.35
LCK P06239 1/20 0.35
PDGFRA P16234 1/20 0.35
PARP1 P09874 2/20 0.31
TNKS2 Q9H2K2 2/20 0.31
PARP2 Q9UGN5 2/20 0.31
TLK2 Q86UE8 1/20 0.31
MEN1 O00255 1/20 0.31
RGS12 O14924 1/20 0.31
NPC1 O15118 1/20 0.31
GMNN O75496 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6088248 0.84 KDR (0.39) KDRPDGFRBSRCFGFR1PKN1
SCHEMBL6088068 0.84 KDR (0.54) KDRPDGFRBSRCFGFR1RET
SCHEMBL6088072 0.84 KDR (0.54) KDRPDGFRBSRCFGFR1RET
SCHEMBL6091270 0.76 KDR (0.40) KDRPDGFRBSRCFGFR1PKN1
SCHEMBL6091525 0.75 LRRK2 (0.36) KDRLRRK2TLK2
SCHEMBL6091530 0.75 LRRK2 (0.36) KDRLRRK2TLK2
SCHEMBL6090793 0.74 KDR (0.46) KDRPDGFRBSRCFGFR1PKN1
SCHEMBL6088365 0.73 KDR (0.47) KDRPDGFRBSRCFGFR1PKN1
SCHEMBL6090489 0.73 KDR (0.43) KDRPDGFRBSRCFGFR1PKN1
SCHEMBL6088285 0.72 KDR (0.46) KDRPDGFRBSRCFGFR1PKN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed