SCHEMBL6089665

SCHEMBL6089665

COCCOCOc1cccc(OCCOc2ccccn2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.41
HTR1A P08908 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
TSHR P16473 3/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
GRM5 P41594 1/20 0.39
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165449 0.81 TSHR (0.44) HTR1AADRA1DADRA1AADRA1BTSHR
SCHEMBL29784889 0.81 TSHR (0.44) HTR1AADRA1DADRA1AADRA1BTSHR
SCHEMBL22297588 0.79 KDM4E (0.52) MAPK1TSHRCYP1A2CYP2D6CYP2C19
SCHEMBL16668774 0.77 TSHR (0.55) MAPK1TSHRCYP1A2CYP2D6CYP2C19
SCHEMBL7520673 0.77 ALDH1A1 (0.52) MAPK1TSHRCYP1A2CYP2D6CYP2C19
SCHEMBL9369921 0.75 KCNA3 (0.50) CYP1A2CYP2C19ALDH1A1MAPTRAB9A
SCHEMBL15723552 0.75 MAPK1 (0.58) MAPK1TSHRCYP1A2CYP2D6CYP2C19
SCHEMBL6089615 0.74 ABCB1 (0.46) HTR1AALDH1A1MAPTRAB9A
SCHEMBL6091732 0.74 CHRNB2 (0.51) HTR1AADRA1DADRA1AADRA1BCYP2D6
SCHEMBL27333271 0.74 NPC1 (0.44) MAPK1HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed