SCHEMBL6089417

SCHEMBL6089417

CCOC(=O)c1c(C=C2C(=O)NN=C2c2cnccn2)[nH]c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.52
CHEK1 O14757 1/20 0.49
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 2/20 0.40
ABL1 P00519 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
FLT3 P36888 1/20 0.40
ALK Q9UM73 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
NPC1 O15118 1/20 0.40
PDE5A O76074 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6089402 1.00 KDR (0.52) KDRCHEK1KDM4EALDH1A1ABL1
SCHEMBL6089795 0.87 KDR (0.42) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6089787 0.87 KDR (0.42) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6088717 0.83 ABL1 (0.40) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6088711 0.83 ABL1 (0.40) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6090600 0.83 KDR (0.61) KDRCHEK1KDM4EALDH1A1ABL1
SCHEMBL6090612 0.83 KDR (0.61) KDRCHEK1KDM4EALDH1A1ABL1
SCHEMBL6089434 0.82 ADORA2B (0.48) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6089440 0.82 ADORA2B (0.48) KDRKDM4EALDH1A1ABL1RET
SCHEMBL6089001 0.81 ABL1 (0.45) KDRKDM4EALDH1A1ABL1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed