SCHEMBL6089903

SCHEMBL6089903

COc1ccc(NC(=O)CC2=NNC(=O)C2=Cc2c[nH]c3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
LMNA P02545 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 3/20 0.46
NTRK1 P04629 4/20 0.46
FLT3 P36888 3/20 0.46
PRKD3 O94806 2/20 0.46
ABL1 P00519 2/20 0.46
RET P07949 2/20 0.46
PDGFRB P09619 2/20 0.46
LTK P29376 2/20 0.46
KDR P35968 2/20 0.46
CSNK1A1 P48729 2/20 0.46
CDK7 P50613 2/20 0.46
MAP2K1 Q02750 2/20 0.46
MST1R Q04912 2/20 0.46
NTRK3 Q16288 2/20 0.46
NTRK2 Q16620 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6089647 0.88 NTRK1 (0.45) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6089642 0.88 NTRK1 (0.45) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6090008 0.82 NTRK1 (0.48) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6088944 0.82 NTRK1 (0.48) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6088938 0.82 NTRK1 (0.48) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6090009 0.82 NTRK1 (0.48) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6091507 0.81 NTRK1 (0.48) ALDH1A1LMNAKDM4EMEN1KMT2A
SCHEMBL6092121 0.80 FLT3 (0.62) ALDH1A1MEN1KMT2AMAPTFLT3
SCHEMBL6092116 0.80 FLT3 (0.62) ALDH1A1MEN1KMT2AMAPTFLT3
SCHEMBL6088227 0.80 CASP3 (0.51) ALDH1A1LMNAKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP claimed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO claimed
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP disclosed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed