SCHEMBL6090145

SCHEMBL6090145

O=C1NN=C(CCc2ccc(O)cc2)C1=Cc1cc(Br)c[nH]1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.34
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
PKM P14618 1/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
LTA4H P09960 1/20 0.31
PDGFRB P09619 1/20 0.31
FGFR1 P11362 1/20 0.31
KDR P35968 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
HTT P42858 1/20 0.30
EGFR P00533 1/20 0.30
MAP4K1 Q92918 1/20 0.30
ERCC1 P07992 1/20 0.30
ERCC4 Q92889 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6090999 0.89 GFER (0.32) MAP4K1
SCHEMBL6090481 0.88 DAO (0.35) PKMKDRGPR84MAP4K1
SCHEMBL6090485 0.88 DAO (0.35) PKMKDRGPR84MAP4K1
SCHEMBL6089530 0.86 PDPK1 (0.34) PDPK1ESR1ESR2LTA4HGPR84
SCHEMBL6089536 0.86 PDPK1 (0.34) PDPK1ESR1ESR2LTA4HGPR84
SCHEMBL6090443 0.80 PDPK1 (0.45) PDPK1PDGFRBFGFR1KDR
SCHEMBL6091331 0.79 CA12 (0.39) PDPK1ESR1ESR2KDRHTT
SCHEMBL6091332 0.79 CA12 (0.39) PDPK1ESR1ESR2KDRHTT
SCHEMBL6091365 0.77 ESR1 (0.33) PDPK1ESR1ESR2GPR84EGFR
SCHEMBL6088593 0.75 GFER (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed