SCHEMBL6091572

SCHEMBL6091572

O=c1ccc2cnc(OCCCCN3CCN(c4nccc5ccc(F)cc45)CC3)nc2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.58
DRD2 P14416 7/20 0.58
HTR2A P28223 7/20 0.58
SLC6A4 P31645 2/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6102727 0.88 HTR1A (0.56) HTR1ADRD2HTR2ASLC6A4
SCHEMBL6091955 0.87 HTR1A (0.44) HTR1ADRD2HTR2ASLC6A4
SCHEMBL4757893 0.86 DRD2 (0.70) HTR1ADRD2HTR2ASLC6A4KCNH2
SCHEMBL6101800 0.82 HTR1A (0.56) HTR1ADRD2HTR2ASLC6A4KCNH2
SCHEMBL5372211 0.78 HTR1A (0.75) HTR1ADRD2HTR2ASLC6A4KCNH2
SCHEMBL6102378 0.77 DRD2 (0.58) HTR1ADRD2HTR2ASLC6A4
SCHEMBL6105551 0.76 HTR1A (0.55) HTR1ADRD2HTR2ASLC6A4
SCHEMBL6103440 0.76 DRD2 (0.61) HTR1ADRD2HTR2ASLC6A4
SCHEMBL5373960 0.76 DRD2 (0.72) HTR1ADRD2HTR2ASLC6A4KCNH2
SCHEMBL5366589 0.75 DRD2 (0.68) HTR1ADRD2HTR2ASLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006090272-A1 ISOQUINOLINE [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2006-08-31 WO claimed
WO-2006090272-A1 ISOQUINOLINE [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2006-08-31 WO disclosed