SCHEMBL6091612

SCHEMBL6091612

O=Cc1[nH]c2ccccc2c1CN1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
ERN1 O75460 1/20 0.51
MAPT P10636 5/20 0.46
ALOX15 P16050 2/20 0.46
PARP1 P09874 1/20 0.46
TSHR P16473 1/20 0.46
KDM4E B2RXH2 3/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 4/20 0.46
GAA P10253 3/20 0.46
HTT P42858 1/20 0.45
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
DRD3 P35462 2/20 0.44
CHRNA7 P36544 1/20 0.44
CYP2A13 Q16696 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14560414 0.87 HTR2A (0.49) ALDH1A1KMT2AMEN1ERN1MAPT
SCHEMBL18886833 0.77 HSD17B10 (0.70) ALDH1A1KMT2AMEN1MAPTALOX15
SCHEMBL31025920 0.77 HSD17B10 (0.70) ALDH1A1KMT2AMEN1MAPTALOX15
SCHEMBL14280374 0.74 KMT2A (1.00) ALDH1A1KMT2AMEN1ERN1MAPT
SCHEMBL29422865 0.74 KMT2A (1.00) ALDH1A1KMT2AMEN1ERN1MAPT
SCHEMBL3282288 0.72 ALDH1A1 (0.60) ALDH1A1MAPTALOX15TSHRKDM4E
SCHEMBL29637659 0.71 MAPT (0.43) ALDH1A1MAPTTSHRKDM4EHPGD
SCHEMBL29956788 0.71 HTT (0.51) ALDH1A1MAPTTSHRKDM4EHPGD
SCHEMBL7380422 0.71 HTT (0.51) ALDH1A1MAPTTSHRKDM4EHPGD
SCHEMBL18886849 0.70 ALDH1A1 (0.53) ALDH1A1KMT2AMEN1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed
EP-1218373-A2 2-PYRAZOLIN-5-ONES AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-07-03 EP disclosed
WO-2001009121-A2 2-PYRAZOLIN-5-ONES_AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed