SCHEMBL6092145

SCHEMBL6092145

O=C(Nc1ccc(NCCN2CCOCC2)nc1)c1c[nH]c2c1C(=O)CCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.40
MAPK14 Q16539 1/20 0.40
MERTK Q12866 2/20 0.39
FYN P06241 2/20 0.38
MELK Q14680 1/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
LMNA P02545 1/20 0.37
KDR P35968 1/20 0.37
SYK P43405 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
KCNH2 Q12809 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
EPHX2 P34913 1/20 0.36
PARP1 P09874 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092785 0.93 KIT (0.41) HPGDKCNH2
SCHEMBL6092075 0.84 HCAR3 (0.40) LMNA
SCHEMBL6095310 0.82 HCAR3 (0.42) MERTKLMNA
SCHEMBL6093483 0.82 HCAR3 (0.43)
SCHEMBL6095908 0.79 HCAR3 (0.41)
SCHEMBL6093985 0.79 ROCK2 (0.35) MELK
SCHEMBL6394774 0.79 ROCK2 (0.42) LMNACYP2C9
SCHEMBL6093234 0.78 KMT2A (0.46) MAPK14LMNAKDRCYP3A4CYP2C9
SCHEMBL6092453 0.77 HTR2C (0.44)
SCHEMBL6092190 0.76 BUB1 (0.47) ALOX15LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109351-B1 Fused pyrrolecarboxamides; GABA brain receptor ligands NEUROGEN CORPORATION (US) 2006-09-19 US disclosed