SCHEMBL6098833

SCHEMBL6098833

CS(=O)(=O)O.CS(=O)(=O)O.C[n+]1ccn(CC2CC(n3cc[n+](C)c3)CN2c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.37

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.33
ALDH1A1 P00352 7/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 4/20 0.31
KMT2A Q03164 4/20 0.31
HTT P42858 1/20 0.30
SIRT6 Q8N6T7 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6098826 0.95 MEN1 (0.33) MAPTALDH1A1MEN1KMT2ASIRT6
SCHEMBL6097562 0.87
SCHEMBL6097556 0.83
SCHEMBL6097660 0.79
Hydrochloric Acid SCHEMBL6098054 0.78
SCHEMBL6096181 0.74 MAPT (0.40) MAPTALDH1A1SMN1; SMN2MEN1KMT2A
Hydrochloric Acid SCHEMBL6097678 0.74 GAA (0.33)
Hydrochloric Acid SCHEMBL6095180 0.74 MAPT (0.39) MAPTALDH1A1MEN1KMT2ASIRT6
SCHEMBL6158539 0.71 MEN1 (0.44) MAPTALDH1A1MEN1KMT2ASIRT6
SCHEMBL6331162 0.71 MEN1 (0.44) MAPTALDH1A1MEN1KMT2ASIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7132543-B2 Para-phenylenediamine derivatives containing a disubstituted pyrrolidinyl group bearing a cationic radical, and use of the same for dyeing keratin fibers L'OREAL S.A. (FR) 2006-11-07 US disclosed
US-20040248961-A1 Para-phenylenediamine derivatives containing a disubstituted pyrrolidinyl group bearing a cationic radical, and use of the same for dyeing keratin fibers L'OREAL S.A. (FR) 2004-12-09 US disclosed
EP-1462453-A1 Paraphenylenediamin derivatives comprising a substituted pyrrolidinyl group and bearing a cationic radical as well as their use for dyeing keratinic fibres L'OREAL (FR) 2004-09-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248961-A1 Para-phenylenediamine derivatives containing a disubstituted pyrrolidinyl group bearing a cationic radical, and use of the same for dyeing keratin fibers KRT18, CDC73, PKN1 MAPT 2722/4885ALDH1A1 783/4885SMN1; SMN2 4204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.