SCHEMBL6100609

SCHEMBL6100609

O=C(O)CC(NC(=O)c1cc(-c2ccc(F)c(Cl)c2)ccc1O)c1ccc(-c2cccc(OC(F)(F)F)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.48
MME P08473 1/20 0.47
P2RX1 P51575 1/20 0.45
DCAF1 Q9Y4B6 1/20 0.45
CTSA P10619 7/20 0.44
DHODH Q02127 1/20 0.43
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43
SUCNR1 Q9BXA5 2/20 0.42
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
MCHR1 Q99705 1/20 0.41
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
FFAR1 O14842 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5926193 0.91 P2RX1 (0.43) MMP12MMEP2RX1DCAF1CTSA
SCHEMBL4827815 0.89 DCAF1 (0.54) MMP12DCAF1CTSASUCNR1
SCHEMBL6100717 0.88 MME (0.49) MMP12MMECTSAITGB3ITGAV
SCHEMBL5927615 0.88 CTSA (0.47) MMEP2RX1DCAF1CTSASUCNR1
SCHEMBL6098336 0.86 MMP12 (0.60) MMP12MMECTSASUCNR1ITGB3
SCHEMBL6100601 0.86 ITGB1 (0.52) MMEP2RX1DHODHTHRATHRB
SCHEMBL3989530 0.85 CTSA (0.48) P2RX1DCAF1CTSAFFAR1
SCHEMBL6097139 0.85 CTSA (0.48) P2RX1DCAF1CTSAFFAR1
SCHEMBL4824692 0.83 MME (0.46) MMEP2RX1DHODHTHRATHRB
SCHEMBL4824688 0.83 MME (0.46) MMEP2RX1DHODHTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122580-B2 Aryl and heteroaryl compounds and methods to modulate coagulation TRANSTECH PHARMA, INC. (US) 2006-10-17 US disclosed