SCHEMBL6103173

SCHEMBL6103173

Cc1cc2cc(F)ccc2c(N2CCN(CCCCOc3ccc4ccc(=O)[nH]c4n3)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 19/20 0.54
HTR1A P08908 18/20 0.54
HTR2A P28223 18/20 0.54
SLC6A4 P31645 7/20 0.43
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6105551 0.94 HTR1A (0.55) DRD2HTR1AHTR2ASLC6A4DRD4
SCHEMBL6101535 0.89 DRD2 (0.59) DRD2HTR1AHTR2ASLC6A4DRD4
SCHEMBL6101800 0.88 HTR1A (0.56) DRD2HTR1AHTR2ASLC6A4KCNH2
SCHEMBL6102727 0.83 HTR1A (0.56) DRD2HTR1AHTR2ASLC6A4
SCHEMBL5373877 0.83 HTR1A (0.68) DRD2HTR1AHTR2ASLC6A4KCNH2
SCHEMBL6104010 0.81 DRD2 (0.72) DRD2HTR1AHTR2A
SCHEMBL5369417 0.81 HTR1A (0.64) DRD2HTR1AHTR2ASLC6A4DRD3
SCHEMBL5364650 0.81 DRD2 (0.72) DRD2HTR1AHTR2ASLC6A4DRD4
SCHEMBL5371781 0.80 DRD2 (0.69) DRD2HTR1AHTR2ASLC6A4DRD4
SCHEMBL5374936 0.79 DRD2 (0.66) DRD2HTR1AHTR2ASLC6A4DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006090272-A1 ISOQUINOLINE [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2006-08-31 WO claimed
WO-2006090272-A1 ISOQUINOLINE [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2006-08-31 WO disclosed