5-Fluorodeoxyuridylate

5-Fluorodeoxyuridylate

SCHEMBL6107

O=c1[nH]c(=O)n([C@H]2C[C@H](O)[C@@H](COP(=O)(O)O)O2)cc1F

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.71
SMN1; SMN2 Q16637 1/20 0.71
TYMS P04818 5/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Fluorodeoxyuridylate SCHEMBL973436 1.00 LMNA (0.71) LMNASMN1; SMN2TYMS
5-Fluorodeoxyuridylate SCHEMBL17117772 1.00 LMNA (0.71) LMNASMN1; SMN2TYMS
5-Fluorodeoxyuridylate SCHEMBL21901970 1.00 LMNA (0.71) LMNASMN1; SMN2TYMS
5-Fluorodeoxyuridylate SCHEMBL15189164 1.00 LMNA (0.71) LMNASMN1; SMN2TYMS
SCHEMBL5491971 0.93 LMNA (0.67) LMNASMN1; SMN2TYMS
SCHEMBL13026822 0.93 LMNA (0.67) LMNASMN1; SMN2TYMS
5-Fluorodeoxyuridylate SCHEMBL15671694 0.92 TYMS (0.64) LMNASMN1; SMN2TYMS
SCHEMBL28378385 0.92 LMNA (0.66) LMNASMN1; SMN2TYMS
5-Fluorodeoxyuridylate SCHEMBL25223991 0.91 LMNA (0.69) LMNASMN1; SMN2TYMS
SCHEMBL5491976 0.91 LMNA (0.69) LMNASMN1; SMN2TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3461 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090505-A1 FLUOROPYRIMIDINE PARTICLES FOR THE TREATMENT OF CANCER WAKE FOREST UNIVERSITY HEALTH SCIENCES (US) 2026-04-30 WO claimed
US-20250360157-A1 CYTOTOXIC FLUOROPYRIMIDINE POLYMERS AND METHODS OF USE THEREOF Wake Forest Univesity Health Sciences (US) 2025-11-27 US claimed
US-20250262215-A1 USE OF CYCLIN E1 STATUS AS A PREDICTIVE BIOMARKER FOR TREATING CANCER WITH WEE1 INHIBITORS ZENO MANAGEMENT, INC. 2025-08-21 US claimed
US-20250262214-A1 INTERMITTENT DOSING REGIMEN FOR AZENOSERTIB IN TREATING CANCER ZENO MANAGEMENT, INC. 2025-08-21 US claimed
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug QINGDAO HAIJI BIOMEDICINE CO., LTD. (CN) 2025-07-22 US claimed
US-20250205217-A1 METHODS OF IMPROVING CANCER IMMUNOTHERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-06-26 US claimed
US-12319915-B2 Cytotoxic fluoropyrimidine polymers and methods of use thereof WAKE FOREST UNIVERSITY HEALTH SCIENCES (US) 2025-06-03 US claimed
CN-119744179-A Conjugates for targeted therapy 梁碧惠 2025-04-01 CN claimed
US-20250059301-A1 Fusion Protein Construct NORTHWESTERN UNIVERSITY 2025-02-20 US claimed
EP-4504267-A1 CONJUGATE FOR TARGETING THERAPY National Taiwan University (TW) 2025-02-12 EP claimed
WO-2003068223-A1 ARYL UREAS WITH RAF KINASE AND ANGIOGENESIS INHIBITING ACTIVITY BAYER CORPORATION (US) 2003-08-21 WO claimed
WO-2003068746-A1 ARYL UREAS AS KINASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-08-21 WO claimed
WO-2003068229-A1 PYRIDINE, QUINOLINE, AND ISOQUINOLINE N-OXIDES AS KINASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-08-21 WO claimed
WO-2003055489-A1 2,4-DIAMINO-PYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003055890-A1 THIENOPYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003040141-A1 OXAZOLYL-PHENYL-2,4-DIAMINO-PYRIMIDINE COMPOUNDS AND METHODS FOR TREATING HYPERPROLIFERATIVE DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2003-05-15 WO claimed
US-5663321-A INHIBITOR OF THYMIDYLATE SYNTHASE; ANTICANCER/ANTITUMOR AGENTS THE BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 1997-09-02 US claimed
US-5614505-A 5-FLUOROURIDINE OR 5-FLUORODEOXYURIDINE, DRUG DELIVERY, IMPROVED BIOAVAILABILITY, ANTICARCINOGENIC AGENTS THE BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 1997-03-25 US claimed
US-5457187-A Antitumor, anticarcinogeic agents BOARD OF REGENTS UNIVERSITY OF NEBRASKA (US) 1995-10-10 US claimed