SCHEMBL6110282

SCHEMBL6110282

Cc1nc(-c2ccco2)nc2sc(C(N)=O)c(N)c12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.68
LIMK1 P53667 3/20 0.59
MAPT P10636 4/20 0.56
HTT P42858 2/20 0.56
USP2 O75604 1/20 0.56
PTK2B Q14289 1/20 0.56
HSD17B10 Q99714 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
RECQL P46063 1/20 0.56
MCL1 Q07820 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
EEF2K O00418 7/20 0.55
KMT2A Q03164 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1176458 0.81 IKBKB (0.68) IKBKBLIMK1MAPTHTTUSP2
SCHEMBL4198561 0.81 IKBKB (1.00) IKBKBLIMK1MAPTHTTUSP2
SCHEMBL6110291 0.80 KMT2A (0.71) IKBKBLIMK1MAPTHTTNPC1
SCHEMBL5026165 0.79 LIMK1 (0.60) IKBKBLIMK1MAPTHTTUSP2
SCHEMBL6111195 0.79 IKBKB (0.56) IKBKBLIMK1MAPTHTTNPC1
SCHEMBL1175798 0.78 IKBKB (0.64) IKBKBLIMK1MAPTHTTUSP2
SCHEMBL6111409 0.78 IKBKB (0.64) IKBKBLIMK1MAPTHTTL3MBTL1
SCHEMBL6111218 0.77 IKBKB (0.66) IKBKBLIMK1MAPTHTTHSD17B10
SCHEMBL1176286 0.77 IKBKB (0.62) IKBKBLIMK1MAPTHTTUSP2
SCHEMBL6111488 0.76 EEF2K (0.59) IKBKBLIMK1MAPTHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006010568-A2 SUBSTITUTED PYRIDO[3',2':4,5]THIENO[3,2-D]PYRIMIDINE-2,4(1 H,3H)-DIONES AND -4(3H)-ONES, PYRIDO[3',2':4,5]FURO[3,2-D]PYRIMIDINE-2,4(1 H,3H)-DIONES AND -4(3H)-ONES, AND USE THEREOF AS INHIBITORS OF TNF-ALPHA RELEASE CURACYTE DISCOVERY GMBH (DE) 2006-02-02 WO disclosed