SCHEMBL6120874

SCHEMBL6120874

CNC(=O)c1c(-c2ccc(Cl)cc2)nn2cc(NS(=O)(=O)CCc3ccc(Br)c(F)c3)c(C3CC3)cc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.36
PTGES2 Q9H7Z7 7/20 0.35
WDR5 P61964 2/20 0.34
SCN7A Q01118 1/20 0.33
SCN5A Q14524 1/20 0.33
RIPK2 O43353 1/20 0.32
ABCB11 O95342 1/20 0.32
EGFR P00533 1/20 0.32
KRAS P01116 1/20 0.32
RAF1 P04049 1/20 0.32
PGR P06401 1/20 0.32
RET P07949 1/20 0.32
CHRM2 P08172 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ARAF P10398 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
FECH P22830 1/20 0.32
KDR P35968 1/20 0.32
MAP2K2 P36507 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6121823 0.94 CYP3A4 (0.36) BRAFPTGES2WDR5CYP2C19CYP3A4
SCHEMBL6121078 0.93 PTGES2 (0.35) BRAFPTGES2WDR5
SCHEMBL6120989 0.92 BRAF (0.34) BRAFPTGES2WDR5CYP2C19CYP3A4
SCHEMBL6120670 0.92 PTGES2 (0.37) BRAFPTGES2WDR5SCN7ASCN5A
SCHEMBL6121300 0.91 PTGES2 (0.38) BRAFPTGES2EGFR
SCHEMBL6120967 0.90 WDR5 (0.36) BRAFPTGES2WDR5CYP2C19CYP3A4
SCHEMBL6120931 0.90 BRAF (0.35) BRAFPTGES2SCN7ASCN5ARIPK2
SCHEMBL6120639 0.89 WDR5 (0.37) BRAFPTGES2WDR5RIPK2ABCB11
SCHEMBL6120536 0.88 BRAF (0.38) BRAFWDR5CHRM1
SCHEMBL6120643 0.88 BRAF (0.34) BRAFPTGES2WDR5CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067664-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed