SCHEMBL6120967

SCHEMBL6120967

CNC(=O)c1c(-c2ccc(F)cc2)nn2cc(NS(=O)(=O)CCc3ccc(Br)c(Cl)c3)c(C3CC3)cc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 2/20 0.36
PTGES2 Q9H7Z7 8/20 0.34
BRAF P15056 4/20 0.33
CYP2C9 P11712 4/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2C19 P33261 3/20 0.33
KCNH2 Q12809 2/20 0.33
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6121078 0.94 PTGES2 (0.35) WDR5PTGES2BRAF
SCHEMBL6121823 0.93 CYP3A4 (0.36) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6120643 0.92 BRAF (0.34) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6120657 0.91 PTGES2 (0.37) PTGES2BRAFJAK2
SCHEMBL6120874 0.90 BRAF (0.36) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6121195 0.89 BRAF (0.32) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6121013 0.87 WDR5 (0.37) WDR5BRAFCYP2C9CYP3A4CYP2C19
SCHEMBL6121734 0.87 CYP2C9 (0.33) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6120989 0.86 BRAF (0.34) WDR5PTGES2BRAFCYP2C9CYP3A4
SCHEMBL6121072 0.86 MAPT (0.36) BRAFCYP2C9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067664-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed