SCHEMBL6125818

SCHEMBL6125818

FCCNN1Cc2ccc(Br)cc2C1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 3/20 0.38
NAMPT P43490 2/20 0.36
PNMT P11086 2/20 0.36
HSD17B3 P37058 4/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
CARM1 Q86X55 2/20 0.35
PRMT5 O14744 2/20 0.34
METAP1 P53582 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145007 0.73 CARM1 (0.42) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL15983781 0.66 HSD17B3 (0.41) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL1782140 0.66 BRD4 (0.46) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL18782916 0.66 DPP8 (0.43) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL578240 0.66 HSD17B3 (0.55) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL16126838 0.66 ABHD6 (0.46) ABHD6NAMPTPNMTHSD17B3DPP8
Bromide SCHEMBL14921932 0.65 DPP8 (0.42) ABHD6NAMPTPNMTHSD17B3DPP8
Hydrochloric Acid SCHEMBL7487148 0.65 CYP19A1 (0.36) ABHD6NAMPTHSD17B3DPP8DPP9
SCHEMBL31197682 0.64 ABHD6 (0.44) ABHD6NAMPTPNMTHSD17B3DPP8
SCHEMBL24502687 0.62 MAOB (0.45) ABHD6HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2640366-A2 BENZOXAZEPINES AS INHIBITORS OF PI3K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE Exelixis, Inc. (US) 2013-09-25 EP disclosed
WO-2012068096-A2 BENZOXAZEPINES AS INHIBITORS OF PI3K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-24 WO disclosed