SCHEMBL6130100

SCHEMBL6130100

CCCCCCCCc1ccc(C(CC(C)(COCc2ccccc2)NC(=O)OCc2ccccc2)OP(=O)(OCc2ccccc2)OCc2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CETP P11597 3/20 0.39
AAK1 Q2M2I8 2/20 0.38
TLR2 O60603 2/20 0.38
MBOAT4 Q96T53 1/20 0.38
PLK1 P53350 3/20 0.37
PLK3 Q9H4B4 3/20 0.37
SMPD1 P17405 1/20 0.35
HDAC1 Q13547 1/20 0.35
S1PR4 O95977 2/20 0.35
S1PR1 P21453 2/20 0.35
S1PR3 Q99500 2/20 0.35
S1PR5 Q9H228 2/20 0.35
S1PR2 O95136 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6130094 0.78 CETP (0.43) CETPTLR2MBOAT4PLK1PLK3
SCHEMBL7620622 0.77 CETP (0.39) CETPTLR2MBOAT4PLK1PLK3
SCHEMBL6130148 0.75 MBOAT4 (0.43) AAK1MBOAT4PLK1PLK3
SCHEMBL6130115 0.72 S1PR1 (0.49) CETPMBOAT4S1PR4S1PR1S1PR3
SCHEMBL6130099 0.72 CETP (0.45) CETPMBOAT4PLK1PLK3S1PR4
Butane SCHEMBL6130095 0.72 S1PR1 (0.48) CETPMBOAT4S1PR4S1PR1S1PR3
SCHEMBL6130104 0.71 SPHK2 (0.42) MBOAT4PLK1PLK3SMPD1S1PR4
SCHEMBL6130097 0.70 CETP (0.42) CETPMBOAT4PLK1PLK3SMPD1
SCHEMBL23944942 0.69 MBOAT4 (0.56) CETPAAK1MBOAT4
SCHEMBL23318030 0.69 MBOAT4 (0.55) CETPMBOAT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1315735-A4 PHOSPHATE DERIVATIVES AS IMMUNOREGULATORY AGENTS MERCK & CO INC (US) 2005-04-06 EP disclosed
EP-1315735-A1 PHOSPHATE DERIVATIVES AS IMMUNOREGULATORY AGENTS Merck & Co., Inc. (US) 2003-06-04 EP disclosed
WO-2002018395-A1 PHOSPHATE DERIVATIVES AS IMMUNOREGULATORY AGENTS MERCK & CO., INC. (US) 2002-03-07 WO disclosed