Laudanosine

Laudanosine

SCHEMBL6130845

COc1ccc(C[C@@H]2c3cc(OC)c(OC)cc3CCN2C)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 1.00
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
HSD17B10 Q99714 2/20 1.00
MAPK1 P28482 1/20 1.00
CYP2D6 P10635 1/20 1.00
ALOX15 P16050 1/20 0.79
DRD2 P14416 1/20 0.76
DRD1 P21728 1/20 0.76
KCNH2 Q12809 2/20 0.71
BCHE P06276 1/20 0.71
ACHE P22303 1/20 0.71
KCNN1 Q92952 1/20 0.67
KCNN2 Q9H2S1 1/20 0.67
KCNN3 Q9UGI6 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Laudanosine SCHEMBL466528 1.00 LMNA (1.00) LMNAKDM4EALDH1A1HSD17B10MAPK1
Laudanosine SCHEMBL30816021 1.00 LMNA (1.00) LMNAKDM4EALDH1A1HSD17B10MAPK1
Laudanosine SCHEMBL466529 1.00 LMNA (1.00) LMNAKDM4EALDH1A1HSD17B10MAPK1
Laudanosine SCHEMBL29822950 1.00 LMNA (1.00) LMNAKDM4EALDH1A1HSD17B10MAPK1
Laudanosine SCHEMBL11398962 0.96 LMNA (0.93) LMNAKDM4EALDH1A1HSD17B10MAPK1
SCHEMBL21346112 0.96 LMNA (0.93) LMNAKDM4EALDH1A1HSD17B10MAPK1
Laudanosine SCHEMBL11398960 0.96 LMNA (0.93) LMNAKDM4EALDH1A1HSD17B10MAPK1
SCHEMBL21346139 0.95 LMNA (0.90) LMNAKDM4EALDH1A1HSD17B10MAPK1
SCHEMBL21346180 0.95 LMNA (0.90) LMNAKDM4EALDH1A1HSD17B10MAPK1
Dimethylgrisabine SCHEMBL30735570 0.92 LMNA (0.84) LMNAKDM4EALDH1A1HSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023086696-A2 APPARATUS AND METHODS FOR CONTINUOUS FLOW SYNTHESIS OF CISATRACURIUM ODH IP Corp. (US) 2023-05-19 WO disclosed
CN-107778234-B Preparation method of neuromuscular blocker intermediate 四川科瑞德制药股份有限公司 2023-01-06 CN disclosed
US-20110185796-A1 CISATRACURIUM DERIVATIVES, PREPARATION AND USES THEREOF CHEMAGIS LTD. (IL) 2011-08-04 US disclosed
WO-2009133556-A2 CISATRACURIUM DERIVATIVES, PREPARATION AND USES THEREOF CHEMAGIS LTD. (IL) 2009-11-05 WO disclosed
EP-0971898-B1 SUBSTITUTED ISOQUINOLINES AS ULTRA SHORT ACTING NEUROMUSCULAR BLOCKERS AVERA PHARMACEUTICALS INC (US) 2005-05-11 EP disclosed
EP-1526130-A1 Substituted isoquinolines as ultra short acting neuromuscular blockers Avera Pharmaceuticals, Inc. (US) 2005-04-27 EP disclosed
US-6177445-B1 MUSCLE RELAXANTS GLAXO WELLCOME INC. 2001-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110185796-A1 CISATRACURIUM DERIVATIVES, PREPARATION AND USES THEREOF CHRNA5, GAP43, CHRNA3 LMNA 1771/4885KDM4E 2186/4885ALDH1A1 2216/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.