SCHEMBL6131857

SCHEMBL6131857

COc1ccc(C=O)cc1OCC#N

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.64
TSHR P16473 1/20 0.64
FDPS P14324 1/20 0.59
LMNA P02545 4/20 0.56
MAPT P10636 4/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
HTT P42858 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
AOX1 Q06278 1/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TRIM24 O15164 1/20 0.50
HPGD P15428 1/20 0.50
ALDH5A1 P51649 1/20 0.50
ABAT P80404 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TRIM33 Q9UPN9 1/20 0.50
PDCD1 Q15116 1/20 0.49
CD274 Q9NZQ7 1/20 0.49
TTR P02766 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433948 0.84 ALDH1A1 (0.64) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL2843898 0.83 ALDH1A1 (0.62) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL2841230 0.82 ALDH1A1 (0.60) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL7661907 0.82 FDPS (0.86) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL5974454 0.80 FDPS (0.77) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL754958 0.80 ALDH1A1 (0.72) ALDH1A1TSHRFDPSLMNAMAPT
SCHEMBL30416638 0.80 ALDH1A1 (0.72) ALDH1A1TSHRFDPSLMNAMAPT
3,4-Dimethoxybenzaldehyde SCHEMBL25202 0.79 ALDH1A1 (1.00) ALDH1A1TSHRFDPSLMNAMAPT
3,4-Dimethoxybenzaldehyde SCHEMBL5308959 0.79 ALDH1A1 (1.00) ALDH1A1TSHRFDPSLMNAMAPT
3,4-Dimethoxybenzaldehyde SCHEMBL1330962 0.79 ALDH1A1 (1.00) ALDH1A1TSHRFDPSLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
US-6479495-B1 SIMULTANEOUSLY TREATING DEPRESSION AND MEMORY DYSFUNCTION IN MAMMALS SUFFERING FROM MEMORY DYSFUNCTION AND DEPRESSION AVENTIS PHARMACEUTICALS INC. 2002-11-12 US disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed