SCHEMBL6131874

SCHEMBL6131874

CNC(=O)Oc1ccc(CCN2CCN(c3ccccc3Cl)CC2)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 4/20 0.57
ADRA1A P35348 4/20 0.57
ADRA1B P35368 4/20 0.57
DRD3 P35462 2/20 0.55
DRD2 P14416 2/20 0.55
DRD4 P21917 1/20 0.55
FAAH O00519 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HTR1A P08908 3/20 0.49
EBP Q15125 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
TMEM97 Q5BJF2 1/20 0.49
HTR2A P28223 2/20 0.49
ADORA2B P29275 1/20 0.48
HTR4 Q13639 1/20 0.48
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
HTR2C P28335 1/20 0.48
HTR7 P34969 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131928 0.90 ADRA1D (0.57) ADRA1DADRA1AADRA1BDRD3DRD2
SCHEMBL6131799 0.89 ADRA1D (0.56) ADRA1DADRA1AADRA1BMEN1KMT2A
SCHEMBL6131869 0.89 ADRA1D (0.60) ADRA1DADRA1AADRA1BDRD3DRD2
Hydrochloric Acid SCHEMBL6132049 0.89 ADRA1D (0.55) ADRA1DADRA1AADRA1BDRD3DRD2
SCHEMBL6131790 0.88 ADRA1D (0.57) ADRA1DADRA1AADRA1BDRD3DRD2
SCHEMBL6132007 0.88 ADRA1D (0.76) ADRA1DADRA1AADRA1BKMT2AHTR1A
SCHEMBL6131894 0.87 ADRA1D (0.53) ADRA1DADRA1AADRA1BDRD3FAAH
Mefeclorazine SCHEMBL2110367 0.86 ADRA1D (0.73) ADRA1DADRA1AADRA1BDRD3DRD2
SCHEMBL6131943 0.82 KDM4E (0.63) DRD3DRD2DRD4KMT2AHTR1A
SCHEMBL6131787 0.81 ADRA1D (0.59) ADRA1DADRA1AADRA1BDRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed