SCHEMBL6132005

SCHEMBL6132005

C#CCOc1cccc(CN2CCc3cc(OC)c(OC)cc3C2)c1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.59
TSHR P16473 2/20 0.59
MAPT P10636 2/20 0.59
KMT2A Q03164 1/20 0.51
DRD3 P35462 3/20 0.49
ALDH1A1 P00352 2/20 0.49
ALOX15 P16050 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
HSD17B10 Q99714 1/20 0.49
POLB P06746 1/20 0.49
PDE4B Q07343 1/20 0.48
ABCB1 P08183 5/20 0.48
DHFR P00374 1/20 0.48
REV1 Q9UBZ9 1/20 0.47
DRD2 P14416 2/20 0.47
DRD1 P21728 2/20 0.47
DRD4 P21917 2/20 0.47
DRD5 P21918 2/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3322960 0.88 KDM4E (0.71) KDM4ETSHRMAPTKMT2ADRD3
Hydrochloric Acid SCHEMBL3320118 0.86 KDM4E (0.70) KDM4ETSHRMAPTKMT2ADRD3
SCHEMBL3049241 0.80 DRD3 (0.71) KDM4ETSHRMAPTDRD3DRD2
SCHEMBL3059563 0.80 REV1 (0.66) KDM4ETSHRMAPTKMT2ADRD3
SCHEMBL6132003 0.79 KDM4E (0.64) KDM4ETSHRMAPTKMT2AALDH1A1
Hydrochloric Acid SCHEMBL6132039 0.78 KDM4E (0.63) KDM4ETSHRMAPTKMT2AALDH1A1
SCHEMBL3058767 0.76 KDM4E (0.55) KDM4ETSHRMAPTKMT2ADRD3
SCHEMBL10753092 0.76 POLB (0.62) KDM4ETSHRMAPTKMT2ADRD3
SCHEMBL3041492 0.76 CA9 (0.69) KDM4ETSHRMAPTKMT2ADRD3
SCHEMBL3324219 0.74 KDM4E (0.63) KDM4ETSHRMAPTKMT2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed