SCHEMBL6132003

SCHEMBL6132003

C#CCOc1cc(CN2CCc3cc(OC)c(OC)cc3C2)ccc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
TDP1 Q9NUW8 1/20 0.64
KMT2A Q03164 1/20 0.60
MAPT P10636 3/20 0.58
GAA P10253 1/20 0.58
RAB9A P51151 1/20 0.58
ABCB1 P08183 7/20 0.58
ABCC1 P33527 4/20 0.58
ABCG2 Q9UNQ0 2/20 0.58
DRD2 P14416 1/20 0.56
REV1 Q9UBZ9 1/20 0.55
DHCR7 Q9UBM7 1/20 0.54
PDE4B Q07343 1/20 0.53
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
TSHR P16473 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6132039 0.99 KDM4E (0.63) KDM4ETDP1KMT2AMAPTGAA
SCHEMBL5667128 0.82 DRD2 (0.65) KDM4EKMT2AMAPTRAB9ADRD2
SCHEMBL3059243 0.82 REV1 (0.78) KDM4ETDP1KMT2AMAPTGAA
SCHEMBL7680831 0.82 DRD2 (0.64) KDM4EKMT2AGAARAB9ADRD2
Hydrochloric Acid SCHEMBL5667186 0.81 DRD2 (0.64) KDM4EKMT2AMAPTRAB9ADRD2
SCHEMBL3059412 0.81 KDM4E (0.86) KDM4ETDP1KMT2AMAPTGAA
Hydrochloric Acid SCHEMBL6132064 0.81 DRD2 (0.63) KDM4EKMT2AGAARAB9ADRD2
SCHEMBL6131905 0.81 DRD2 (0.63) KDM4EKMT2AGAADRD2ALDH1A1
Bromide SCHEMBL6132084 0.80 DRD2 (0.61) KDM4EKMT2AGAADRD2ALDH1A1
SCHEMBL6132005 0.79 KDM4E (0.59) KDM4ETDP1KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed