SCHEMBL6132050

SCHEMBL6132050

COc1cc(CN2CCc3cc(OC)c(OC)cc3C2)ccc1O

nearest known ligand 0.82

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 10/20 0.82
KDM4E B2RXH2 3/20 0.81
TDP1 Q9NUW8 1/20 0.81
PDE4B Q07343 1/20 0.79
MAPT P10636 2/20 0.79
ALDH1A1 P00352 1/20 0.79
HTT P42858 1/20 0.79
NPSR1 Q6W5P4 1/20 0.79
TAAR1 Q96RJ0 1/20 0.79
GAA P10253 1/20 0.74
RAB9A P51151 1/20 0.74
ABCC1 P33527 5/20 0.71
ABCG2 Q9UNQ0 2/20 0.71
CA2 P00918 1/20 0.71
CA9 Q16790 1/20 0.71
KMT2A Q03164 1/20 0.68
DHCR7 Q9UBM7 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416542 0.96 KDM4E (0.79) ABCB1KDM4ETDP1PDE4BMAPT
SCHEMBL3059412 0.92 KDM4E (0.86) ABCB1KDM4ETDP1PDE4BMAPT
SCHEMBL29836069 0.88 KDM4E (0.93) ABCB1KDM4ETDP1PDE4BMAPT
SCHEMBL3059315 0.85 ABCB1 (0.77) ABCB1KDM4ETDP1PDE4BMAPT
SCHEMBL3810641 0.84 KMT2A (0.76) ABCB1KDM4ETDP1MAPTGAA
SCHEMBL3051392 0.83 CA2 (0.73) ABCB1KDM4ETDP1MAPTALDH1A1
SCHEMBL3506177 0.83 CA2 (0.73) ABCB1KDM4ETDP1MAPTALDH1A1
SCHEMBL30760754 0.83 ABCB1 (1.00) ABCB1KDM4ETDP1ABCC1ABCG2
SCHEMBL5131462 0.83 KDM4E (0.71) ABCB1KDM4ETDP1MAPTALDH1A1
SCHEMBL3050097 0.83 CA9 (1.00) ABCB1KDM4ETDP1PDE4BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed