SCHEMBL6136003

SCHEMBL6136003

O=C(O)Cc1cccc(NC(=O)Nc2ccccc2)c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 1/20 0.78
SELP P16109 2/20 0.60
SELE P16581 2/20 0.60
EPHX2 P34913 2/20 0.59
TP53 P04637 1/20 0.59
EPHX1 P07099 1/20 0.59
TSHR P16473 1/20 0.59
CDK9 P50750 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
CLK4 Q9HAZ1 1/20 0.59
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
NR1H4 Q96RI1 2/20 0.57
NPC1 O15118 1/20 0.57
LMNA P02545 1/20 0.57
MAPT P10636 1/20 0.57
HTT P42858 1/20 0.57
RAB9A P51151 1/20 0.57
MGLL Q99685 1/20 0.56
SELL P14151 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30557308 1.00 HPSE (0.78) HPSESELPSELEEPHX2TP53
SCHEMBL11628807 0.87 HPSE (0.65) HPSESELPSELESMN1; SMN2MEN1
SCHEMBL7387069 0.85 DDX3X (0.71) HPSEMEN1KMT2ANR1H4NPC1
SCHEMBL7251772 0.85 RAB9A (0.66) HPSESELPSELESMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL11628069 0.85 HPSE (0.63) HPSESELPSELESMN1; SMN2MEN1
SCHEMBL30802742 0.84 SMN1; SMN2 (0.61) HPSEEPHX2TP53EPHX1TSHR
SCHEMBL27954484 0.84 SMN1; SMN2 (0.61) HPSEEPHX2TP53EPHX1TSHR
SCHEMBL11630238 0.84 HPSE (0.62) HPSESELPSELESMN1; SMN2MEN1
SCHEMBL5151866 0.84 KMT2A (0.74) HPSEEPHX2TP53EPHX1TSHR
SCHEMBL11628800 0.84 HPSE (0.61) HPSESELPSELEEPHX1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042279-B1 SUBSTITUTED BETA-ALANINES AVENTIS PHARMA LTD (GB) 2005-03-02 EP disclosed
US-6352977-B1 ALANINE WITH PRODRUGS AVENTIS PHARMA LIMITED (GB) 2002-03-05 US disclosed
EP-1042279-A1 SUBSTITUTED BETA-ALANINES Aventis Pharma Limited (GB) 2000-10-11 EP disclosed
WO-1999033789-A1 SUBSTITUTED β-ALANINES AVENTIS PHARMA LIMITED (GB) 1999-07-08 WO disclosed