SCHEMBL6137705

SCHEMBL6137705

O=C(O)c1c(Cl)ccc2[nH]cnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.48
PARP1 P09874 2/20 0.42
ACLY P53396 1/20 0.42
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
ALK Q9UM73 3/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
LMNA P02545 2/20 0.39
DPP8 Q6V1X1 1/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38
AURKA O14965 2/20 0.37
DAPK3 O43293 2/20 0.37
PRKD3 O94806 2/20 0.37
MAP4K4 O95819 2/20 0.37
RET P07949 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6137870 0.81 NR4A2 (0.40) PARP1ACLYEGLN1LMNAPOLB
SCHEMBL10713217 0.81 PARP1 (0.47) DPP4PARP1ACLYKDM5AKDM4C
SCHEMBL13544495 0.79 PARP1 (0.42) DPP4PARP1ACLYALDH1A1KDM4E
SCHEMBL29894129 0.79 PARP1 (0.42) DPP4PARP1ACLYALDH1A1KDM4E
SCHEMBL24754415 0.77 SMN1; SMN2 (0.39) PARP1ACLYKDM5AKDM4EEGLN1
SCHEMBL1080823 0.77 PARP1 (0.41) DPP4PARP1ALDH1A1KDM4EHSD17B10
SCHEMBL1081560 0.76 CA12 (0.47) DPP4PARP1ALDH1A1KDM4EEGLN1
SCHEMBL1081796 0.76 EGLN1 (0.46) DPP4PARP1ACLYKDM4CALDH1A1
SCHEMBL4535246 0.74 DPP4 (0.44) DPP4PARP1ACLYALKALDH1A1
SCHEMBL6137724 0.72 POLB (0.36) DPP4PARP1ACLYALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515956-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM (US) 2005-08-10 EP disclosed
EP-1515956-A1 PEPTIDE DEFORMYLASE INHIBITORS Smithkline Beecham (US) 2005-03-23 EP disclosed
WO-2003104209-A1 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-12-18 WO disclosed