SCHEMBL6137870

SCHEMBL6137870

COC(=O)c1c(Cl)ccc2[nH]cnc12

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.40
ALOX5 P09917 3/20 0.39
POLB P06746 1/20 0.39
LMNA P02545 3/20 0.39
PARP1 P09874 1/20 0.39
NOTUM Q6P988 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
ACLY P53396 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
EGLN1 Q9GZT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6137724 0.90 POLB (0.36) NR4A2ALOX5POLBLMNAPARP1
SCHEMBL21986865 0.83 LMNA (0.40) NR4A2POLBLMNAPARP1SMN1; SMN2
SCHEMBL1081543 0.82 LMNA (0.39) NR4A2ALOX5POLBLMNAPARP1
SCHEMBL1080724 0.82 QPCT (0.44) POLBLMNAPARP1
SCHEMBL24754415 0.81 SMN1; SMN2 (0.39) PARP1SMN1; SMN2ACLYEGLN1
SCHEMBL6137705 0.81 DPP4 (0.48) POLBLMNAPARP1ACLYGAA
SCHEMBL1081831 0.79 ALDH1A1 (0.40) NR4A2POLBLMNAPARP1EGLN1
SCHEMBL6137875 0.76 MKNK1 (0.39) NR4A2POLBLMNANOTUMSMN1; SMN2
SCHEMBL11022639 0.76 ALPL (0.41) NR4A2ALOX5POLBLMNAGAA
SCHEMBL22533838 0.73 PARP1 (0.42) NR4A2PARP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4499630-A1 BCL-XL INHIBITORS BeiGene, Ltd. (KY) 2025-02-05 EP disclosed
US-20250034128-A1 BCL-XL INHIBITORS BEIGENE, LTD. (KY) 2025-01-30 US disclosed
CN-118974033-A Bcl-xL inhibitors 百济神州有限公司 2024-11-15 CN disclosed
WO-2023185986-A1 BCL-XL INHIBITORS BEIGENE , LTD. (KY) 2023-10-05 WO disclosed
EP-1515956-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM (US) 2005-08-10 EP disclosed
EP-1515956-A1 PEPTIDE DEFORMYLASE INHIBITORS Smithkline Beecham (US) 2005-03-23 EP disclosed
WO-2003104209-A1 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250034128-A1 BCL-XL INHIBITORS BCL2, BCL2L1, BCL2L10 NR4A2 2528/4885ALOX5 2330/4885POLB 1598/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.