SCHEMBL6138350

SCHEMBL6138350

O=C(O)C1(N2CCCC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.38
HSD11B1 P28845 3/20 0.37
HSD11B2 P80365 1/20 0.37
HTT P42858 1/20 0.33
FFAR3 O14843 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15194218 0.97 ALDH1A1 (0.38) ALDH1A1TP53TSHRHSD11B1HSD11B2
SCHEMBL234076 0.97 ALDH1A1 (0.41) ALDH1A1TP53TSHRHSD11B1HSD11B2
Hydrochloric Acid SCHEMBL15194272 0.95 ALDH1A1 (0.40) ALDH1A1TP53TSHRHSD11B1HSD11B2
Hydrochloric Acid SCHEMBL15194419 0.95 ALDH1A1 (0.40) ALDH1A1TP53TSHRHSD11B1HSD11B2
SCHEMBL5332707 0.92 ALDH1A1 (0.38) ALDH1A1TP53TSHRHSD11B1HSD11B2
SCHEMBL14858388 0.90 ALDH1A1 (0.40) ALDH1A1TP53TSHRHSD11B1HSD11B2
SCHEMBL14061763 0.90 KDM1A (0.35) ALDH1A1TP53TSHRHSD11B1HSD11B2
SCHEMBL5323192 0.89
SCHEMBL25435115 0.87 ALDH1A1 (0.38) ALDH1A1TP53TSHRHTTFFAR3
SCHEMBL5569331 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013120921-A9 NOVEL PYRROLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2015-10-08 WO disclosed
EP-2814822-A1 NOVEL PYRROLIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2014-12-24 EP disclosed
WO-2013120921-A1 NOVEL PYRROLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2013-08-22 WO disclosed
EP-1170281-B1 1,1- and 1,2-disubstituted cyclopropanes, process for their preparation and pharmaceutical compositions thereof SERVIER LAB (FR) 2005-12-21 EP disclosed
EP-1170281-A1 1,1- and 1,2-disubstituted cyclopropanes, process for their preparation and pharmaceutical compositions thereof LES LABORATOIRES SERVIER (FR) 2002-01-09 EP disclosed