SCHEMBL6138536

SCHEMBL6138536

CCOC(=O)CN(C)CCC(/C=C/c1ccccc1OCCCCCc1ccccc1)Cc1ccc(C(=O)O)c(C)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.44
PDE4B Q07343 3/20 0.44
PDE4C Q08493 3/20 0.44
PDE4D Q08499 3/20 0.44
LTA4H P09960 3/20 0.43
S1PR1 P21453 2/20 0.36
RARB P10826 1/20 0.36
ALOX5 P09917 2/20 0.34
PPARG P37231 2/20 0.34
PTGES O14684 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
RXRA P19793 1/20 0.33
LTB4R Q15722 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
CXCR2 P25025 1/20 0.33
ABCB1 P08183 1/20 0.33
PPARA Q07869 1/20 0.33
AKR1C3 P42330 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3598408 0.87 LTA4H (0.44) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL3598346 0.87 LTA4H (0.44) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL3598347 0.87 LTA4H (0.44) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL3593691 0.84 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL6138195 0.84 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL3593694 0.84 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL3595599 0.82 LTA4H (0.42) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL3595602 0.82 LTA4H (0.42) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL3595606 0.82 LTA4H (0.42) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL6138471 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216223-B1 NOVEL DICARBOXYLIC ACID DERIVATIVES WITH PHARMACEUTICAL PROPERTIES BAYER HEALTHCARE AG (DE) 2005-11-09 EP disclosed
EP-1216223-A1 NOVEL DICARBOXYLIC ACID DERIVATIVES WITH PHARMACEUTICAL PROPERTIES Bayer Aktiengesellschaft (DE) 2002-06-26 EP disclosed
WO-2001019778-A1 NOVEL DICARBOXYLIC ACID DERIVATIVES WITH PHARMACEUTICAL PROPERTIES BAYER AKTIENGESELLSCHAFT (DE) 2001-03-22 WO disclosed