SCHEMBL6139004

SCHEMBL6139004

COc1ccc(CN2CCN(c3cc(N4CCCC4)nc(N4CCCC4)n3)CC2)c(OCCCCCCC(=O)O)c1OC

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 7/20 0.46
KMT2A Q03164 7/20 0.46
LMNA P02545 2/20 0.46
CASP1 P29466 6/20 0.46
CASP5 P51878 6/20 0.46
CASP4 P49662 5/20 0.46
MGLL Q99685 1/20 0.44
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6774817 0.99 KDM4E (0.46) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL6139052 0.97 KDM4E (0.49) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6772881 0.96 KDM4E (0.48) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6778734 0.89 ALDH1A1 (0.44) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6774850 0.86 ALDH1A1 (0.45) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6771210 0.85 MEN1 (0.57) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6772490 0.83 MEN1 (0.59) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6778263 0.81 LMNA (0.55) KDM4EALDH1A1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6774183 0.80 MEN1 (0.62) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL6138665 0.80 KDM4E (0.68) KDM4EALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1277746-B1 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions thereof SERVIER LAB (FR) 2005-05-11 EP disclosed
EP-1277746-A2 N-benzylpiperazine derivatives, process for their preparation and pharmaceutical compositions thereof Les Laboratoires Servier (FR) 2003-01-22 EP disclosed