SCHEMBL6139775

SCHEMBL6139775

CC(=O)c1ccc(-c2ccc(F)cc2)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.51
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SRD5A2 P31213 2/20 0.46
FASN P49327 1/20 0.46
SYK P43405 1/20 0.45
HSD17B1 P14061 3/20 0.45
PTGS2 P35354 1/20 0.44
PRKAB2 O43741 1/20 0.44
PRKAG1 P54619 1/20 0.44
PRKAA2 P54646 1/20 0.44
PRKAA1 Q13131 1/20 0.44
PRKAG3 Q9UGI9 1/20 0.44
PRKAG2 Q9UGJ0 1/20 0.44
PRKAB1 Q9Y478 1/20 0.44
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11585221 0.90 HSD17B1 (0.54) PTGS1KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL7367792 0.83 MAPT (0.55) KMT2AMEN1KDM4EALDH1A1SMN1; SMN2
SCHEMBL11540874 0.83 PTGS1 (0.54) PTGS1KMT2AMEN1KDM4EALDH1A1
SCHEMBL27467828 0.83 MAPT (0.44) KMT2AMEN1ALDH1A1SMN1; SMN2SRD5A2
SCHEMBL16156050 0.81 PTGS1 (0.53) PTGS1KMT2AMEN1KDM4EALDH1A1
SCHEMBL11540045 0.80 PTGS1 (0.51) PTGS1KMT2AMEN1KDM4EALDH1A1
SCHEMBL1226198 0.79 PTGS1 (0.54) PTGS1KMT2AMEN1KDM4EALDH1A1
SCHEMBL30837198 0.79 SRD5A2 (0.66) KMT2AMEN1KDM4ESMN1; SMN2SRD5A2
SCHEMBL16492515 0.79 SRD5A2 (0.66) KMT2AMEN1KDM4ESMN1; SMN2SRD5A2
SCHEMBL6139808 0.79 PTGS1 (0.43) PTGS1KMT2AMEN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196403-B1 ANTIPSYCHOTIC CYCLIC N-ARALKYL AMINES SANOFI AVENTIS (FR) 2005-11-09 EP disclosed
US-6908914-B1 Antipsychotic cyclic N-aralkylamines SANOFI-SYNTHELABO (FR) 2005-06-21 US disclosed
EP-1192122-B1 BENZENE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI SYNTHELABO (FR) 2003-10-22 EP disclosed
US-6482986-B1 Benzene derivatives, preparation method and pharmaceutical compositions containing same SANOFI-SYNTHELABO (FR) 2002-11-19 US disclosed
EP-1196403-A1 ANTIPSYCHOTIC CYCLIC N-ARALKYL AMINES Sanofi-Aventis (FR) 2002-04-17 EP disclosed
EP-1192122-A1 BENZENE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-04-03 EP disclosed
WO-2001002380-A1 ANTIPSYCHOTIC CYCLIC N-ARALKYL AMINES SANOFI-SYNTHELABO (FR) 2001-01-11 WO disclosed
WO-2000076953-A1 BENZENE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2000-12-21 WO disclosed