SCHEMBL6139875

SCHEMBL6139875

NC1=Nc2cc(CCCNCc3cccc(Cl)c3)ccc2C2CCCC12F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 12/20 1.00
NOS1 P29475 12/20 1.00
NOS2 P35228 11/20 1.00
CHRM2 P08172 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
OPRM1 P35372 1/20 0.35
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6137653 0.99 NOS1 (0.98) NOS3NOS1NOS2CHRM2CYP1A2
SCHEMBL6137346 0.79 NOS3 (0.66) NOS3NOS1NOS2CHRM2CYP1A2
Hydrochloric Acid SCHEMBL7174141 0.78 NOS3 (0.64) NOS3NOS1NOS2
SCHEMBL6137320 0.72 NOS3 (1.00) NOS3NOS1NOS2
SCHEMBL6561325 0.71 NOS1 (0.98) NOS3NOS1NOS2CHRM2CYP1A2
Hydrochloric Acid SCHEMBL6069276 0.71 NOS1 (1.00) NOS3NOS1NOS2CHRM2CYP1A2
SCHEMBL6137615 0.69 NOS3 (0.68) NOS3NOS1NOS2
SCHEMBL6137654 0.69 NOS3 (0.68) NOS3NOS1NOS2
SCHEMBL6137311 0.68 NOS1 (1.00) NOS3NOS1NOS2
SCHEMBL6561433 0.67 NOS1 (0.98) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129077-B9 FLUORINATED 3,4-DIHYDROQUINOLINE DERIVATIVES USED AS NOS INHIBITORS SCHERING AG (DE) 2005-07-20 EP claimed
EP-1129077-B1 FLUORINATED 3,4-DIHYDROQUINOLINE DERIVATIVES USED AS NOS INHIBITORS SCHERING AG (DE) 2005-04-20 EP claimed