SCHEMBL6139976

SCHEMBL6139976

O=C(O)CC(NC(=O)C1(c2ccc(Cl)cc2)CCCC1)c1ccc2nc(-c3ccccc3[N+](=O)[O-])ccc2c1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSA P10619 10/20 0.40
MAPT P10636 4/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PSMD14 O00487 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC4 P56524 1/20 0.34
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3318102 0.84 ITGB1 (0.45)
SCHEMBL3317824 0.69 ITGA4 (0.61)
SCHEMBL3313019 0.69 ITGB1 (0.47) TRPA1
SCHEMBL5173387 0.68 ITGB1 (0.44) MEN1KMT2AL3MBTL1HDAC4
SCHEMBL3316847 0.68 ITGB1 (0.48)
SCHEMBL3313181 0.66 ITGB1 (0.66)
SCHEMBL4625262 0.66 ITGB1 (0.66)
SCHEMBL3315803 0.66 ALDH1A1 (0.37) MAPTMEN1KMT2AL3MBTL1HDAC4
SCHEMBL4624848 0.65 ITGB1 (0.54)
SCHEMBL4626449 0.65 ITGB1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed